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Found 32 from University of Bergen
TargetMyeloblastin(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-cobratoxin(Naja kaouthia)
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50554678(CHEMBL4779503)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of TAMRA-HAKTYMWDGWYMPTSH-NH2 from Naja kaouthia alpha-cobratoxin by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50156156(2-Amino-7-(1,2-dihydroxy-propyl)-5,6,7,8-tetrahydr...)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity for human phenylalanine hydroxylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-cobratoxin(Naja kaouthia)
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50554679(CHEMBL4740171)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of TAMRA-HAKTYMWDGWYMPTSH-NH2 from Naja kaouthia alpha-cobratoxin by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50:  530nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylalanine-4-hydroxylase(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50156156(2-Amino-7-(1,2-dihydroxy-propyl)-5,6,7,8-tetrahydr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against human phenylalanine hydroxylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50031631(CHEMBL3359767)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50171289(Benzenemethanesulfonyl fluoride | CHEMBL190503 | P...)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-cobratoxin(Naja kaouthia)
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50554678(CHEMBL4779503)
Affinity DataIC50:  2.90E+4nMAssay Description:Displacement of TAMRA-HAKTYMWDGWYMPTSH-NH2 from Naja kaouthia alpha-cobratoxin by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207528(CHEMBL3925060)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207531(CHEMBL3897010)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207532(CHEMBL3939235)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207533(CHEMBL3956669)
Affinity DataEC50:  6.17E+4nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207531(CHEMBL3897010)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207534(CHEMBL3957870)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207533(CHEMBL3956669)
Affinity DataEC50:  6.10E+4nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207536(CHEMBL3929127)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207537(CHEMBL3911275)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207536(CHEMBL3929127)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207534(CHEMBL3957870)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207538(CHEMBL3931202)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207535(CHEMBL3902257)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207529(CHEMBL3933958)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207532(CHEMBL3939235)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207537(CHEMBL3911275)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207538(CHEMBL3931202)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207530(CHEMBL3930236)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207528(CHEMBL3925060)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207529(CHEMBL3933958)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Bergen

Curated by ChEMBL
LigandPNGBDBM50207530(CHEMBL3930236)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity at wild-type human CXCR4 expressed in COS7 cells co-expressing chimeric galphai assessed as inhibition of CXCL12-induced [3H]inos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed